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Peptide Therapy GuideClear peptide education

Understand the source comparison

Neuropeptides Explained Brain Function — Comparison Across Key Peptide Classes

Opioid Peptides (endorphins, enkephalins, dynorphins) Periaqueductal gray, nucleus accumbens, amygdala, spinal cord dorsal horn (MOR), (DOR), (KOR) opioid receptors Pain modulation, reward signaling, stress-induced analgesia, addiction vulnerability Dysr

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  • Opioid Peptides (endorphins, enkephalins, dynorphins)
  • Periaqueductal gray, nucleus accumbens, amygdala, spinal cord dorsal horn
  • μ (MOR), δ (DOR), κ (KOR) opioid receptors
  • Pain modulation, reward signaling, stress-induced analgesia, addiction vulnerability
  • Dysregulation implicated in chronic pain syndromes, opioid use disorder, stress-related psychiatric conditions
  • Most studied neuropeptide system due to clinical relevance. Endogenous opioid tone determines both pain threshold and addiction susceptibility
  • Neuropeptide Y (NPY)
  • Arcuate nucleus, amygdala, hippocampus, cortex
  • Y1, Y2, Y5 receptors
  • Appetite stimulation, anxiety reduction, circadian regulation, stress resilience, memory consolidation
  • Low NPY associated with PTSD, depression, metabolic syndrome; Y2 agonists under investigation for obesity
  • Single most abundant neuropeptide in mammalian brain. Regulates both metabolic homeostasis and emotional resilience through parallel circuits
  • Orexins (Hypocretins A/B)
  • Lateral hypothalamus (exclusive synthesis site)
  • OX1 (Hcrtr1), OX2 (Hcrtr2) receptors
  • Wakefulness stabilization, motivation, reward seeking, autonomic arousal
  • Orexin neuron loss causes narcolepsy; OX2 antagonists (suvorexant) used as sleep aids
  • Orexins link arousal state to motivational salience. Narcolepsy patients lose wakefulness specifically during emotionally charged moments
  • Vasopressin & Oxytocin
  • Paraventricular nucleus, supraoptic nucleus (synthesis); nucleus accumbens, amygdala (release)
  • V1a, V1b, OXTR (oxytocin receptor)
  • Social bonding, trust behavior, aggression, parental care, stress buffering, HPA axis regulation
  • Intranasal oxytocin studied for autism spectrum disorder, social anxiety; vasopressin implicated in aggression, pair bonding
  • Differ by only two amino acids but produce opposite effects on aggression and affiliation. Receptor distribution determines behavioral output
  • Tachykinins (Substance P, Neurokinin A/B)
  • Dorsal horn of spinal cord, amygdala, striatum, cortex
  • NK1, NK2, NK3 receptors
  • Pain amplification, anxiety, emesis, inflammatory modulation, neurogenic inflammation
  • NK1 antagonists developed for chemotherapy-induced nausea; substance P implicated in fibromyalgia, IBS
  • Substance P amplifies glutamate signaling at NMDA receptors. Blocking NK1 reduces pain without analgesic tolerance typical of opioids